WitrynaTheranostic approaches with adrenal specific radiotracers hold promise for improved diagnostics and treatment. Here, we report a new theranostic approach to advanced … The majority of the new compounds inhibited cortisol and aldosterone secretion in a dose-dependent manner both NCI-H295 cells and Y1 cells transfected with either human CYP11B1 or CYP11B2, indicating target enzyme binding. The IC50 values for inhibition of cortisol and aldosterone in Y1 cells are … Zobacz więcej The metabolic stability of [125I]IMTO and three new tracers was determined by radio-HPLC; results are listed in Table 2. The esters 3 and 4 exhibited nearly equal or even better … Zobacz więcej The intracellular uptake in human adrenocortical NCI-H295 cells was analyzed for [125I]IMTO and the compounds exhibiting the highest metabolic … Zobacz więcej The compounds 3-tetrahydrofurylester 3 and 2,2-difluoroethylester 4 and IMAZA exhibited both strong enzyme inhibition and at least comparable metabolic stability to IMTO, so they were additionally investigated in … Zobacz więcej As both target enzymes are localized at the inner mitochondrial membrane, cellular subfractionation experiments were performed using human NCI-H295 cells. As shown in … Zobacz więcej
"Rekordowa" oferta dla Imaza. Ale i sama Jagiellonia ma wątpliwości
Witryna3 mar 2024 · IMAZA targeting adrenocortical carcinoma; All therapies provide efficacious treatment and only few adverse effects are observed. The preparation of clinical trials … Witrynawspolczesna.pl how many prisons in the united states
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WitrynaThieme E-Books & E-Journals. Full-text search Full-text search; Author Search; Title Search; DOI Search Witryna26 wrz 1990 · Najwyższa wartość rynkowa: 1,50 mln €. 18 sie 2024. Ostatnia zmiana: 30 mar 2024. Wartość rynkowa w szczególe. Nazwisko w kraju pochodzenia: Jesús Imaz Ballesté Data urodzenia: 26 wrz 1990 Miejsce urodzenia: Lleida Wiek: 32 Wzrost: 1,74 m Narodowość: Hiszpania Pozycja: Pomocnik - Ofensywny pomocnik Noga: … Witryna10 kwi 2024 · WPHUB. Jagiellonia Białystok. Wiadomości. Galerie. Wyniki/Kalendarz. Relacje na żywo. Deja vu Jesusa Imaza. Lechia Gdańsk w coraz gorszej sytuacji. Jagiellonia Białystok pokonała 1:0 (0:0 ... how many prisons in south africa